Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ki for monomerid = 50428890
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50428890(ASENAPINE | Saphris)
Affinity DataKi:  0.25nMAssay Description:Antagonist activity at human recombinant 5HT6 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50428890(ASENAPINE | Saphris)
Affinity DataKi:  0.910nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced intracellular calcium release measured fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50428890(ASENAPINE | Saphris)
Affinity DataKi:  2.5nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in HEK293 cells assessed as inhibition of 5HT-induced intracellular calcium release measured fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed