Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ki for monomerid = 8049
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM8049(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 20 | 4...)
Affinity DataKi:  290nM ΔG°:  -37.9kJ/molepH: 7.4 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at 30 °C with substrate, and test compounds in the presence of 100 uM ATP/ [gamma-32P...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Cyclacel

LigandPNGBDBM8049(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 20 | 4...)
Affinity DataKi: >2.00E+4nM ΔG°: >-27.3kJ/moleT: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at 30 °C with substrate, and test compounds in the presence of 100 uM ATP/ [gamma-32P...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed