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Found 1 Enz. Inhib. hit(s) with Target = '11-beta-hydroxysteroid dehydrogenase 1' and Ligand = 'BDBM50339808'
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
University Of Technology

Curated by ChEMBL
LigandPNGBDBM50339808(CHEMBL1689279 | N-[(5aR,7aR,7bS,9aS,12S,13aR,15aR,...)
Affinity DataIC50:  4.50E+4nMAssay Description:Inhibition of human recombinant 11beta-HSD1 expressed in HEK293 cells assessed as conversion of [1,2-[3H]cortisone to cortisol after 10 mins by scint...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed