Found 5 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1A' and Ligand = 'BDBM50241119' Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
King Fahd University Of Petroleum & Minerals
King Fahd University Of Petroleum & Minerals
Affinity DataKi: 7.19nM ΔG°: -48.3kJ/molepH: 7.4 T: 2°CAssay Description:Human-cloned 5-HT1A serotonin receptors stably expressed in HEK293-EBNA cells (Perkin-Elmer, Waltham, MA) were radiolabeled with 1.0nM [3H]-8-OH-DPAT...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
King Fahd University Of Petroleum & Minerals
King Fahd University Of Petroleum & Minerals
Affinity DataKi: 9.30nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor determined using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
King Fahd University Of Petroleum & Minerals
King Fahd University Of Petroleum & Minerals
Affinity DataKi: 9.30nMAssay Description:Agonist activity at 5HT1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Pierre Fabre Research Center
Curated by ChEMBL
Pierre Fabre Research Center
Curated by ChEMBL
Affinity DataKi: 65nMAssay Description:Displacement of [3H]OH-DPAT from rat cortex 5HT1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
King Fahd University Of Petroleum & Minerals
King Fahd University Of Petroleum & Minerals
Affinity DataEC50: 324nMAssay Description:Agonist activity at human 5HT1A receptor in HeLa cells assessed as stimulation of [35S]GTP-gamma-S bindingMore data for this Ligand-Target Pair
