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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1A' and Ligand = 'BDBM50274835'
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute and Karolinska University Hospital

Curated by ChEMBL
LigandPNGBDBM50274835(CHEMBL511857 | trans-1-(4-(3-methoxyphenyl)cyclohe...)
Affinity DataKi:  0.0280nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in human HeLa cell membranes assessed as stimulation of [35S]GTPgammaS binding after 20 mins by l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute and Karolinska University Hospital

Curated by ChEMBL
LigandPNGBDBM50274835(CHEMBL511857 | trans-1-(4-(3-methoxyphenyl)cyclohe...)
Affinity DataEC50:  0.324nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in CHO cells after 90 mins by beta-arrestin-2 recruitment assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Karolinska Institute and Karolinska University Hospital

Curated by ChEMBL
LigandPNGBDBM50274835(CHEMBL511857 | trans-1-(4-(3-methoxyphenyl)cyclohe...)
Affinity DataEC50:  0.794nMAssay Description:Agonist activity at human 5-HT1A receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 15 mins by EL...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed