Found 7 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2C' and Ligand = 'BDBM50108306' Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Texas Health Science Center
Curated by ChEMBL
University Of North Texas Health Science Center
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Texas Health Science Center
Curated by ChEMBL
University Of North Texas Health Science Center
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity against human 5-hydroxytryptamine 2C receptor using displacement of [3H]DOBMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Texas Health Science Center
Curated by ChEMBL
University Of North Texas Health Science Center
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Tested for binding affinity of the compound towards human 5-hydroxytryptamine 2C receptor using [3H]-DOB as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Texas Health Science Center
Curated by ChEMBL
University Of North Texas Health Science Center
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Displacement of [3H]-DOB from human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Texas Health Science Center
Curated by ChEMBL
University Of North Texas Health Science Center
Curated by ChEMBL
Affinity DataKi: 85nMAssay Description:Tested for binding affinity of the compound towards human 5-hydroxytryptamine 2C receptor using [3H]-Mesulergine as radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Texas Health Science Center
Curated by ChEMBL
University Of North Texas Health Science Center
Curated by ChEMBL
Affinity DataKi: 85nMAssay Description:Tested for binding affinity of the compound towards human 5-hydroxytryptamine 2C receptor using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Efficacy (pEC50) was evaluated for 5-HT2C receptor-mediated stimulation of IP3 formation in vitro in choroid plexus of the ratMore data for this Ligand-Target Pair
