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Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 6' and Ligand = 'BDBM50340727'
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Avincuro Pharmaceuticals

US Patent
LigandPNGBDBM50340727(2,5,7-Triimethyl-phenylsulfonyl-pyrazolo[1,5-a]pyr...)
Affinity DataKi:  68.4nM IC50:  147nMAssay Description:Radioligand binding assay using 5-HT6 receptors.More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Avincuro Pharmaceuticals

US Patent
LigandPNGBDBM50340727(2,5,7-Triimethyl-phenylsulfonyl-pyrazolo[1,5-a]pyr...)
Affinity DataKi:  68.4nMAssay Description:Displacement of [3H]lysergic acid diethylamide from human recombinant 5HT6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Avincuro Pharmaceuticals

US Patent
LigandPNGBDBM50340727(2,5,7-Triimethyl-phenylsulfonyl-pyrazolo[1,5-a]pyr...)
Affinity DataKi:  88.8nMAssay Description:Antagonist activity at human recombinant 5HT6 receptor expressed in HEK293 cells assessed as inhibition of serotonin-induced cAMP production after 2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed