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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'A-kinase anchor protein 7 isoform gamma' and Ligand = 'BDBM212603'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
A-kinase anchor protein 7 isoform gamma


(Human)
BDBM212603
PNG
(US9556111, Table 1.7)
Show SMILES OC(=O)c1csc(CN(CCC(c2ccccc2)c2ccccc2)Cc2ccc(F)cc2)n1
Show InChI InChI=1S/C27H25FN2O2S/c28-23-13-11-20(12-14-23)17-30(18-26-29-25(19-33-26)27(31)32)16-15-24(21-7-3-1-4-8-21)22-9-5-2-6-10-22/h1-14,19,24H,15-18H2,(H,31,32)
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/an/an/a 1.80E+4n/an/an/an/a



UNIVERSITETET I OSLO

US Patent


Assay Description
Stable and optimal assay conditions were determined by cross-titrating GST-AKAP18δ and biotinylated PLB using 10 μg/ml glutathione acceptor...


US Patent US9556111 (2017)

More data for this
Ligand-Target Pair