BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Adenomatous polyposis coli protein' and Ligand = 'BDBM270607'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Adenomatous polyposis coli protein


(Homo sapiens (Human))
BDBM270607
PNG
(US10071086, Compound 128)
Show SMILES Fc1ccc(cc1)-c1cncc2[nH]c(nc12)-c1n[nH]c2ncc(cc12)-c1cncc(NC(=O)Cc2ccccc2)c1
Show InChI InChI=1S/C31H19FN8O/c32-22-8-6-19(7-9-22)25-16-34-17-26-28(25)38-31(37-26)29-24-12-21(14-35-30(24)40-39-29)20-11-23(15-33-13-20)36-27(41)10-18-4-2-1-3-5-18/h1-9,11-17H,10H2,(H,36,41)/b31-29+
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 90n/an/an/an/an/an/a



Samumed, LLC

US Patent


Assay Description
Reporter cell lines can be generated by stably transducing cells of cancer cell lines (e.g., colon cancer) with a lentiviral construct that include a...


US Patent US10071086 (2018)

More data for this
Ligand-Target Pair