BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Adenomatous polyposis coli protein' and Ligand = 'BDBM275570'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Adenomatous polyposis coli protein


(Homo sapiens (Human))
BDBM275570
PNG
(US10071086, Compound 547)
Show SMILES CCNCc1cncc(c1)-c1cnc2[nH]nc(-c3nc4c(cccc4[nH]3)-c3cccc(F)c3)c2c1
Show InChI InChI=1S/C27H20FN7/c1-2-29-12-16-9-18(14-30-13-16)19-11-22-25(34-35-26(22)31-15-19)27-32-23-8-4-7-21(24(23)33-27)17-5-3-6-20(28)10-17/h3-11,13-15,29H,2,12H2,1H3/b27-25+
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 97n/an/an/an/an/an/a



Samumed, LLC

US Patent


Assay Description
Reporter cell lines can be generated by stably transducing cells of cancer cell lines (e.g., colon cancer) with a lentiviral construct that include a...


US Patent US10071086 (2018)

More data for this
Ligand-Target Pair