Affinity DataKi: 62nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Binding affinity for Adenosine A1 receptor using N-[3H] cyclohexyladenosine in rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Ability to inhibit binding of [3H]-CHA to adenosine A1 receptor in rat brain cortical membranes.More data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor of rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Binding affinity for Adenosine A1 receptor using N-[3H] cyclohexyladenosine in rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Binding affinity against adenosine A1 receptor from rat forebrain membranes using N6-[3H]-cyclohexyladenosineMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Binding affinity for Adenosine A1 receptor using N-[3H] cyclohexyladenosine in rat forebrain membranes under usual lightMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Tested for binding affinity against Adenosine A1 receptor from rat forebrain membranes, using N6-[3H]- cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 577nMAssay Description:Affinity against Adenosine A1 receptor in rat brain using [3H]- PIA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 930nMAssay Description:Inhibition of [3H]-DPCPX binding to rat cerebral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 930nMAssay Description:Inhibition of [3H]DPCPX binding to adenosine A1 receptor of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Binding affinity against adenosine A1 receptor from guinea pig forebrain membranes, using N6-[3H]-cyclohexyladenosine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Binding affinity against Adenosine A1 receptor from guinea pig forebrain membranes by N6-[3H]- cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Binding affinity for Adenosine A1 receptor using N-[3H] cyclohexyladenosine in guinea pig forebrain membranes under usual lightMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding Affinity towards Adenosine A1 receptor expressed in CHO-K1 cells versus [3H]-CCPAMore data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Inhibitory activity against cyclic AMP production in rat Adenosine A1 receptor assayMore data for this Ligand-Target Pair