TargetAdenosine receptor A1(Rattus norvegicus (rat))
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Ability to inhibit binding of [3H]-CHA to adenosine A1 receptor in rat brain cortical membranes.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranes after 90 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells after 90 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Affinity DataKi: 2.80E+4nMAssay Description:Displacement of [3H]-N6-(2-phenylisopropyl)adenosine from Adenosine A1 receptor in rat cortical membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Affinity DataKi: 2.80E+4nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Affinity DataKi: 2.80E+4nMAssay Description:Ability to inhibit binding of [3H]-R-PIA to Adenosine A1 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Affinity DataKi: 2.82E+4nMAssay Description:Displacement of [3H]-PIA from adenosine A1 receptors of rat brain membraneMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Julius-Maximilians-UniversitäT WüRzburg
Curated by ChEMBL
Affinity DataKi: 2.82E+4nMAssay Description:Affinity against Adenosine A1 receptor in rat brain using [3H]- PIA as radioligandMore data for this Ligand-Target Pair