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Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50205709'
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50205709((2R,3R,4S,5R)-2-(6-amino-2-(phenylethynyl)-9H-puri...)
Affinity DataKi:  391nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50205709((2R,3R,4S,5R)-2-(6-amino-2-(phenylethynyl)-9H-puri...)
Affinity DataKi:  391nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50205709((2R,3R,4S,5R)-2-(6-amino-2-(phenylethynyl)-9H-puri...)
Affinity DataKi:  646nMAssay Description:Displacement [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membrane incubated for 60 mins by microplate beta scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Yamasa Shoyu

Curated by ChEMBL
LigandPNGBDBM50205709((2R,3R,4S,5R)-2-(6-amino-2-(phenylethynyl)-9H-puri...)
Affinity DataKi:  701nMAssay Description:Inhibition of [3H]CHA binding to adenosine A1 receptor from rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed