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Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50316887'
TargetAdenosine receptor A1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50316887(2-amino-8-(2-morpholinoethoxy)-4-phenyl-5H-indeno[...)
Affinity DataKi:  48nMAssay Description:Antagonist activity at human recombinant adenosine A1 receptor by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50316887(2-amino-8-(2-morpholinoethoxy)-4-phenyl-5H-indeno[...)
Affinity DataKi:  48.2nMAssay Description:Antagonistic activity at adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50316887(2-amino-8-(2-morpholinoethoxy)-4-phenyl-5H-indeno[...)
Affinity DataKi:  48.2nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50316887(2-amino-8-(2-morpholinoethoxy)-4-phenyl-5H-indeno[...)
Affinity DataEC50:  48nMAssay Description:Binding affinity to human recombinant adenosine A1 receptor expressed in CHO cells using [3H]CCPA by functional activity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed