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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM97465'
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM97465(US8470800, B | US8609833, 85)
Affinity DataKi:  2.63nMAssay Description:The affinities of selected Purine Derivatives for the adenosine A1 receptor were determined by measuring the displacement of specific [3H] 2-chloro-N...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A1(Homo sapiens (Human))
Inotek Pharmaceuticals

US Patent
LigandPNGBDBM97465(US8470800, B | US8609833, 85)
Affinity DataKi:  2.63nM ΔG°:  -45.5kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assay using adenosine receptor.More data for this Ligand-Target Pair
In DepthDetails US Patent