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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50125910'
TargetAdenosine receptor A2a(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50125910(1-(2-Furan-2-yl-8-methyl-9-methylsulfanyl-8H-pyraz...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]- SCH-58261 binding at human Adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50125910(1-(2-Furan-2-yl-8-methyl-9-methylsulfanyl-8H-pyraz...)
Affinity DataIC50:  17.5nMAssay Description:Antagonist activity as inhibition of cAMP generation after agonist-modulation of human Adenosine A2A receptor with 100 nM NECAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed