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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50257074'
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257074(CHEMBL474016 | N-(2-(4-methoxyphenyl)-1-oxo-1,2-di...)
Affinity DataKi:  4.54nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257074(CHEMBL474016 | N-(2-(4-methoxyphenyl)-1-oxo-1,2-di...)
Affinity DataKi:  4.54nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257074(CHEMBL474016 | N-(2-(4-methoxyphenyl)-1-oxo-1,2-di...)
Affinity DataEC50:  36.3nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in CHO cells assessed as blockade of NECA-mediated inhibition of forskolin-stimulated cA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed