Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]I-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in CHO cells by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair