Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Alpha-1A adrenergic receptor' and Ligand = 'BDBM50063906'
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Merck

Curated by ChEMBL
LigandPNGBDBM50063906((S)-4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-1-(f...)
Affinity DataKi:  580nMAssay Description:Compound was evaluated for its ability to displace [125I]-HEAT binding from rat Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50063906((S)-4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-1-(f...)
Affinity DataKi:  1.70E+3nMAssay Description:Compound was tested for binding affinity utilizing cloned receptor binding assays by using [125 I]HEAT as radioligand to the human Alpha-1A adrenergi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50063906((S)-4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-1-(f...)
Affinity DataIC50:  1.90E+3nMAssay Description:Compound was tested for the tissue binding affinity using [3H]- Prazosin as radioligand to the human prostate Alpha-1A adrenergic receptor subtypeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Merck

Curated by ChEMBL
LigandPNGBDBM50063906((S)-4-(4-Amino-6,7-dimethoxy-quinazolin-2-yl)-1-(f...)
Affinity DataIC50:  2.00E+3nMAssay Description:Compound was tested for the tissue binding affinity using [3H]- Prazosin as radioligand to the rat prostate Alpha-1A adrenergic receptor subtypeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed