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Found 5 Enz. Inhib. hit(s) with Target = 'Alpha-1D adrenergic receptor' and Ligand = 'BDBM50022722'
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50022722((+)2-Amino-1-phenyl-propan-1-ol | (1R, 2R)-2-Amino...)
Affinity DataKi:  8.40E+3nMAssay Description:Binding affinity towards rat cloned Alpha-1D adrenergic receptor ;value ranges from (5.5 -13)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50022722((+)2-Amino-1-phenyl-propan-1-ol | (1R, 2R)-2-Amino...)
Affinity DataKi:  8.51E+3nMAssay Description:In vitro binding affinity towards alpha-1D adrenergic receptor of rat clone in radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50022722((+)2-Amino-1-phenyl-propan-1-ol | (1R, 2R)-2-Amino...)
Affinity DataKi:  8.51E+3nMAssay Description:Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50022722((+)2-Amino-1-phenyl-propan-1-ol | (1R, 2R)-2-Amino...)
Affinity DataEC50:  7.59E+4nMAssay Description:Agonist activity at alpha1D adrenoreceptor in Rattus norvegicus (rat) aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50022722((+)2-Amino-1-phenyl-propan-1-ol | (1R, 2R)-2-Amino...)
Affinity DataEC50:  5.80E+4nMAssay Description:Effective concentration of the compound was determined in vitro against rat aorta Alpha-1D adrenergic receptor;* indicates EC50 < 15% at a concentrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed