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Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-2A adrenergic receptor' and Ligand = 'BDBM50417348'
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417348(CHEMBL1276247)
Affinity DataKi:  166nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50417348(CHEMBL1276247)
Affinity DataEC50:  3.16E+3nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed