Affinity DataKi: 166nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.16E+3nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair