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Found 3 Enz. Inhib. hit(s) with Target = 'Alpha-2A adrenergic receptor' and Ligand = 'BDBM66983'
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
Affinity DataKi:  9.40nMAssay Description:Inhibition of [3H]rauwolscine binding to CHO cells expressing the human Alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(GUINEA PIG)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In DepthDetails PubMed