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Found 4 Enz. Inhib. hit(s) with Target = 'Alpha-2B adrenergic receptor' and Ligand = 'BDBM50412245'
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)
Affinity DataKi:  339nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)
Affinity DataKi:  339nMAssay Description:Binding affinity at human alpha2B ARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)
Affinity DataKi:  339nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenoceptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50412245(CHEMBL495095)
Affinity DataKi:  339nMAssay Description:Displacement of [3H]RS79948-197 from human recombinant adrenergic alpha2B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed