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Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-2C adrenergic receptor' and Ligand = 'BDBM50262235'
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50262235(rilmenidine)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]RX821001 from human alpha2C adrenoceptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50262235(rilmenidine)
Affinity DataKi:  4.68E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed