Affinity DataKi: 1.10nMAssay Description:Displacement of [125I]-[Nle75, Tyr77] Pyr1-apelin-13 from YFP-tagged human APJ receptor expressed in HEK293 cell membranes after 1 hr by gamma-counti...More data for this Ligand-Target Pair
Affinity DataEC50: 272nMAssay Description:Binding affinity against sigma receptor from guinea pig brain (minus cerebellum) homogenates, using [3H]ditolylguanidine (DTG) as radioligand.More data for this Ligand-Target Pair
Affinity DataEC50: 469nMAssay Description:Binding affinity against dopamine receptor D2 from rat striatal homogenates using [3H]YM-09151-2More data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Binding affinity against human bradykinin receptor B2 using [3H]bradykinin as radioligandMore data for this Ligand-Target Pair