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Found 2 Enz. Inhib. hit(s) with Target = 'Apoptosis regulator Bcl-2' and Ligand = 'BDBM50384340'
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50384340(CHEMBL2031009 | US9346795, 328)
Affinity DataIC50:  8.78nMT: 2°CAssay Description:The assays were performed in black flat-bottom 384-well plates. The final assay volume was 50 μl prepared from additions of Gst-Bcl-2 (Bcl-2: GE...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50384340(CHEMBL2031009 | US9346795, 328)
Affinity DataIC50:  9nMAssay Description:Inhibition of GST-tagged Bcl2 using [FAM]-IWIAQELRRIGDEFNAYY-NH2 as substrate after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed