Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Aurora kinase A' and Ligand = 'BDBM36470'
TargetAurora kinase A(Homo sapiens (Human))
Praecis Pharmaceuticals

LigandPNGBDBM36470(2-(4-(3,4-Dimethoxyphenylamino)-6-(quinolin-6-ylam...)
Affinity DataIC50:  270nMpH: 9.5 T: 2°CAssay Description:Selection of DNA-encoded libraries (DELs) which are covalent attachment of encoding double stranded DNA to small-molecule created using a combination...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Praecis Pharmaceuticals

LigandPNGBDBM36470(2-(4-(3,4-Dimethoxyphenylamino)-6-(quinolin-6-ylam...)
Affinity DataIC50:  270nMAssay Description:Inhibition of aurora A kinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Praecis Pharmaceuticals

LigandPNGBDBM36470(2-(4-(3,4-Dimethoxyphenylamino)-6-(quinolin-6-ylam...)
Affinity DataIC50:  270nMAssay Description:Inhibition of aurora A kinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Praecis Pharmaceuticals

LigandPNGBDBM36470(2-(4-(3,4-Dimethoxyphenylamino)-6-(quinolin-6-ylam...)
Affinity DataIC50:  270nMAssay Description:Competitive inhibition of Aurora A by DEL methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed