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Found 2 Enz. Inhib. hit(s) with Target = 'Beta-1 adrenergic receptor' and Ligand = 'BDBM50098661'
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50098661(2-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonyla...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of I-iodocyanopindolol binding to human beta 1 adrenergic receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Wyeth-Ayerst Research

Curated by ChEMBL
LigandPNGBDBM50098661(2-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonyla...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro activity to increase cAMP levels in Chinese hamster ovary (CHO) cells expressing the cloned human beta 1 Adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed