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Found 5 Enz. Inhib. hit(s) with Target = 'Beta-lactamase' and Ligand = 'BDBM50212642'
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212642(CHEMBL70269)
Affinity DataIC50:  2.33nMAssay Description:Tested for the inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
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TargetBeta-lactamase(Staphylococcus aureus)TBA
LigandPNGBDBM50212642(CHEMBL70269)
Affinity DataIC50:  116nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
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TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212642(CHEMBL70269)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
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TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212642(CHEMBL70269)
Affinity DataIC50:  1.46E+4nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
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TargetBeta-lactamase(Enterobacter cloacae)TBA
LigandPNGBDBM50212642(CHEMBL70269)
Affinity DataIC50:  1.84E+4nMAssay Description:Inhibitory activity against Enterobacter cloacae HC8 Class-I beta-lactamase enzyme type P99More data for this Ligand-Target Pair
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