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Found 2 Enz. Inhib. hit(s) with Target = 'Bile salt export pump' and Ligand = 'BDBM78934'
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM78934(2-methoxyacetic acid [(1S,2S)-2-[2-[3-(1H-benzimid...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt export pump(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM78934(2-methoxyacetic acid [(1S,2S)-2-[2-[3-(1H-benzimid...)
Affinity DataIC50:  4.38E+4nMAssay Description:Inhibition of human BSEP overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-taurocholate in presence of ATP measured after 15 to ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed