Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Bombesin receptor subtype-3' and Ligand = 'BDBM50340973'
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50340973((R)-N-(tert-butylcarbamoyl)-4-(quinuclidin-3-ylami...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50340973((R)-N-(tert-butylcarbamoyl)-4-(quinuclidin-3-ylami...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human BRS3 by functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50340973((R)-N-(tert-butylcarbamoyl)-4-(quinuclidin-3-ylami...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse BRS3 by functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed