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Found 4 Enz. Inhib. hit(s) with Target = 'Bombesin receptor subtype-3' and Ligand = 'BDBM50447475'
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447475(CHEMBL3115390)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447475(CHEMBL3115390)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447475(CHEMBL3115390)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447475(CHEMBL3115390)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed