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Found 1 hit Enz. Inhib. hit(s) with Target = 'Bromodomain adjacent to zinc finger domain protein 2B' and Ligand = 'BDBM50148279'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Bromodomain adjacent to zinc finger domain protein 2B


(Homo sapiens (Human))
BDBM50148279
PNG
(CHEMBL3769753)
Show SMILES CC(=O)c1cc(-c2ccc(CO)cc2)c2ccccn12
Show InChI InChI=1S/C17H15NO2/c1-12(20)17-10-15(16-4-2-3-9-18(16)17)14-7-5-13(11-19)6-8-14/h2-10,19H,11H2,1H3
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
GoogleScholar
CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a 4.10E+3n/an/an/an/an/an/a



GlaxoSmithKline

Curated by ChEMBL


Assay Description
Inhibition of recombinant His6-TEV fused human BAZ2B expressed in Escherichia coli incubated for 30 mins in presence of biotinylated peptide by alpha...


J Med Chem 59: 1410-24 (2016)


Article DOI: 10.1021/acs.jmedchem.5b00209
BindingDB Entry DOI: 10.7270/Q2PK0J09
More data for this
Ligand-Target Pair