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Found 2 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM50112344'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50112344(CHEMBL3609314)
Affinity DataKi:  27nMAssay Description:Binding affinity to BRD4 (unknown origin) expressed in Escherichia coli BL21 after 1 hr by proprietary competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50112344(CHEMBL3609314)
Affinity DataIC50:  33nMAssay Description:Displacement of Bio-JQ1 from recombinant human His6 tagged BRD4 bromodomain 1 by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed