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Found 3 Enz. Inhib. hit(s) with Target = 'C-C chemokine receptor type 9' and Ligand = 'BDBM50113430'
TargetC-C chemokine receptor type 9(Homo sapiens (Human))
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50113430(CHEMBL3604499)
Affinity DataIC50:  34nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) assessed as inhibition of TECK-induced calcium mobilization incubated for 10 mins prior to TECK...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 9(Homo sapiens (Human))
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50113430(CHEMBL3604499)
Affinity DataIC50:  34nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by buffer chemotaxis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 9(Homo sapiens (Human))
Cubist Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50113430(CHEMBL3604499)
Affinity DataIC50:  170nMAssay Description:Antagonist activity at CCR9 receptor (unknown origin) by serum chemotaxis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed