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Found 2 Enz. Inhib. hit(s) with Target = 'CREB-binding protein' and Ligand = 'BDBM50178202'
TargetCREB-binding protein(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM50178202(CHEMBL3813701 | US10206931, Example 132)
Affinity DataIC50:  8.62E+3nMAssay Description:His/Flag epitope tagged CBP was cloned, expressed, and purified to homogeneity. CBP binding and inhibition was assessed by monitoring the engagement ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCREB-binding protein(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM50178202(CHEMBL3813701 | US10206931, Example 132)
Affinity DataIC50:  1.20E+5nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP (unknown origin) incubated for 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed