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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM35873'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM35873(5,6-bis(4-chlorophenyl)-N-(piperidin-1-yl)pyrazine...)
Affinity DataIC50:  4nMpH: 7.4 T: 2°CAssay Description:A GTP-gamma-S CB1 functional assay was used to assess the potency of the pyrazine derivatives. [35S]GTP-gamma-S binding assays were performed at 30 d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM35873(5,6-bis(4-chlorophenyl)-N-(piperidin-1-yl)pyrazine...)
Affinity DataIC50:  8.13nMAssay Description:Antagonist activity against human recombinant cannabinoid-1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed