Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50251132'
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251132(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-N-(cyclo...)
Affinity DataIC50:  127nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Sprague-Dawley rat cerebella membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Central Research Institute

Curated by ChEMBL
LigandPNGBDBM50251132(4-((4-Bromophenyl)(2-chlorophenyl)methyl)-N-(cyclo...)
Affinity DataIC50:  146nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHOK1 cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed