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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50040990'
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50040990(CHEMBL3354954)
Affinity DataEC50:  6.70nMAssay Description:Agonist activity at rat recombinant CB2 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50040990(CHEMBL3354954)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed