Affinity DataKi: 47nMAssay Description:Displacement of [3H]CP-55,940 from human CB2 receptor expressed in CHO cell membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 128nMAssay Description:Antagonist activity at human CB2 receptor transfected in CHO cells assessed as inhibition of WIN 55,212-2 mediated suppression of forksolin induced c...More data for this Ligand-Target Pair
Affinity DataEC50: 858nMAssay Description:Inverse agonist activity at human CB2 receptor transfected in CHO cells assessed as increase in forksolin stimulated cAMP production by scintillation...More data for this Ligand-Target Pair