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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50202519'
TargetCannabinoid receptor 2(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50202519(CHEMBL3909238)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50202519(CHEMBL3909238)
Affinity DataIC50:  475nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as reduction in NKH-477-induced intracellular cAMP levels after 30 mins in ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed