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Found 4 Enz. Inhib. hit(s) with Target = 'Carbonic anhydrase 9' and Ligand = 'BDBM50387125'
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Romanian Academy

Curated by ChEMBL
LigandPNGBDBM50387125(4-ureidophenyl sulfamate ring derivative 3j | CHEM...)
Affinity DataKi:  5nMAssay Description:Inhibition of human carbonic anhydrase-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Romanian Academy

Curated by ChEMBL
LigandPNGBDBM50387125(4-ureidophenyl sulfamate ring derivative 3j | CHEM...)
Affinity DataKi:  6nMAssay Description:Inhibition of human recombinant transmembrane CA9 preincubated for 15 mins by stopped-flow CO2 hydration methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Romanian Academy

Curated by ChEMBL
LigandPNGBDBM50387125(4-ureidophenyl sulfamate ring derivative 3j | CHEM...)
Affinity DataKi:  6nMAssay Description:Inhibition of human carbonic anhydrase 9 preincubated for 15 mins measured for 10 to 100 sec using phenol red indicator-based stopped flow assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Romanian Academy

Curated by ChEMBL
LigandPNGBDBM50387125(4-ureidophenyl sulfamate ring derivative 3j | CHEM...)
In DepthDetails ArticlePubMed