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Found 3 Enz. Inhib. hit(s) with Target = 'Cathepsin K' and Ligand = 'BDBM19768'
TargetCathepsin K(Oryctolagus cuniculus (rabbit))
Celera Genomics

Curated by ChEMBL
LigandPNGBDBM19768(Cbz-Leu-NH-CH2-CN | JMC487688 Compound 8 | benzyl ...)
Affinity DataKi:  34.7nMAssay Description:Inhibitory constant against rabbit cathepsin K using Z-Phe-Arg-AMC substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universitat Bonn

LigandPNGBDBM19768(Cbz-Leu-NH-CH2-CN | JMC487688 Compound 8 | benzyl ...)
Affinity DataKi:  35nMAssay Description:Enzyme activities were calculated from kinetic measurements performed by fluorimetric detection of the product AMC at the wavelengths for excitation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universitat Bonn

LigandPNGBDBM19768(Cbz-Leu-NH-CH2-CN | JMC487688 Compound 8 | benzyl ...)
Affinity DataIC50:  39nMAssay Description:The substrate hydrolysis with or without inhibitor was monitored at an excitation wavelength of 360nm and an emission wavelength of 460 nm on a fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed