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Found 3 Enz. Inhib. hit(s) with Target = 'Cholesteryl ester transfer protein' and Ligand = 'BDBM50092197'
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50092197(CHEMBL313006 | S-2-(1-(2-ethylbutyl)cyclohexanecar...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of CETP in human plasma measured every 30 mins for 120 mins by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50092197(CHEMBL313006 | S-2-(1-(2-ethylbutyl)cyclohexanecar...)
Affinity DataIC50:  6.00E+3nMAssay Description:In vitro inhibition of CETP activity was assessed by measuring the rate of [3H]- cholesteryl ester transfer from HDL to apoprotein B-containing lipop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50092197(CHEMBL313006 | S-2-(1-(2-ethylbutyl)cyclohexanecar...)
Affinity DataIC50:  6.00E+3nMAssay Description:In vitro concentration required to inhibit 50% of cholesteryl ester transfer protein mediated cholesteryl ester transfer from HDL to VLDL and LDL in ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed