Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Cholinesterase' and Ligand = 'BDBM50244216'
TargetCholinesterase(Homo sapiens (Human))
University Of Louisiana At Lafayette

Curated by ChEMBL
LigandPNGBDBM50244216(2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-one | CH...)
Affinity DataIC50:  1.78E+4nMAssay Description:Inhibition of BuChE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCholinesterase(Equus caballus (Horse))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50244216(2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-one | CH...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of equine serum BuChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50244216(2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-one | CH...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 10 mins followed by addition of substrate and measured ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Louisiana At Lafayette

Curated by ChEMBL
LigandPNGBDBM50244216(2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-one | CH...)
Affinity DataIC50:  2.51E+4nMAssay Description:Inhibition of BuchE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
University Of Louisiana At Lafayette

Curated by ChEMBL
LigandPNGBDBM50244216(2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-one | CH...)
Affinity DataIC50:  4.51E+4nMAssay Description:Inhibition of human BChE pre-incubated for 6 mins before ATCI substrate addition and measured after 12 mins by DTNB reagent dependent UV-Vis spectrop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed