Found 1 Enz. Inhib. hit(s) with Target = 'Cytochrome P450 2C9' and Ligand = 'BDBM298494'
TargetCytochrome P450 2C9(Homo sapiens (Human)) Boehringer Ingelheim International
US Patent
LigandBDBM298494(US10125101, Example 33 in WO 2013/178575)
Affinity DataIC50: 7.00E+3nMAssay Description:The inhibition of cytochrome P450 2C9-isoenzyme catalyzed hydroxylation of diclofenac by the test compound is assayed at 37° C. with human liver micr...More data for this Ligand-Target Pair