Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'D(1A) dopamine receptor' and Ligand = 'BDBM199158'
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Fudan University

LigandPNGBDBM199158(3,11-dimethoxy-5,6,8,9,14,14a-hexahydrobenzo[4,5]a...)
Affinity DataKi:  5.32nMAssay Description:The transfection of plasmid and membrane preparations was conducted as described in our previous report, with 0.7 nm [3H] SCH23390 (D1R) or [3H]Spipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Fudan University

LigandPNGBDBM199158(3,11-dimethoxy-5,6,8,9,14,14a-hexahydrobenzo[4,5]a...)
Affinity DataKi:  8.80nMAssay Description:The transfection of plasmid and membrane preparations was conducted as described in our previous report, with 0.7 nm [3H] SCH23390 (D1R) or [3H]Spipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Fudan University

LigandPNGBDBM199158(3,11-dimethoxy-5,6,8,9,14,14a-hexahydrobenzo[4,5]a...)
Affinity DataKi:  72.8nMAssay Description:The transfection of plasmid and membrane preparations was conducted as described in our previous report, with 0.7 nm [3H] SCH23390 (D1R) or [3H]Spipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Fudan University

LigandPNGBDBM199158(3,11-dimethoxy-5,6,8,9,14,14a-hexahydrobenzo[4,5]a...)
Affinity DataIC50:  140nMpH: 7.5Assay Description:The [35S]GTPγS binding assay was performed at 30 °C for 30 min containing 10 μgof membrane protein in a final volume of 100 μL with va...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed