TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
Affinity DataKi: 0.0860nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
Affinity DataKi: 0.0900nMAssay Description:Compound was evaluated for the inhibition constant against dopamine receptor D2 in ratMore data for this Ligand-Target Pair
Affinity DataKi: 0.117nMAssay Description:Displacement of [3H]N-methylspiperone from human D2L receptor expressed in HEK293 cell membranes measured after 60 mins by MicroBeta scintillation co...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
Affinity DataKi: 0.120nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
Affinity DataKi: 0.190nMAssay Description:Compound was evaluated for binding affinity towards dopamine receptor D2 in striatal membranes, using [3H]- spiperone as radioligand in the presence ...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
Affinity DataKi: 0.260nMAssay Description:Displacement of [3H]N-methylspiperone from human D2R expressed in HEK293 cell membranes incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
Affinity DataKi: 0.990nMAssay Description:Displacement of [3H]- spiperone from dopamine receptor D2 of striatal membranes without sodium chlorideMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
Affinity DataIC50: 0.920nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal dopamine receptor D2 was determined in vitroMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
Affinity DataIC50: 0.920nMAssay Description:Tested in vitro for inhibition of [3H]spiperone binding to dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
Affinity DataIC50: 0.920nMAssay Description:In vitro ability to inhibit the binding of [3H]spiperone to dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at DRD2 (unknown origin) expressed in HEK293T cells transfected with Galphai1-RLuc8 and gamma2-GFP10 assessed as inhibition of qu...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
Affinity DataKd: 0.170nMAssay Description:Evaluated in vivo for the affinity towards Dopamine receptor D2 of rat striatal tissueMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Washington University
Curated by PDSP Ki Database
Washington University
Curated by PDSP Ki Database
Affinity DataKd: 0.170nMAssay Description:Affinity constant of compound was evaluated in rat striatum tissue preparation.More data for this Ligand-Target Pair