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Found 2 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50216041'
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216041(3-(4-(4-(2-methoxyphenyl)-1-piperazinyl)butyl)quin...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]Spiperone from human Dopamine receptor D2 isoform long expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216041(3-(4-(4-(2-methoxyphenyl)-1-piperazinyl)butyl)quin...)
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human Dopamine receptor D2 isoform long expressed in HEK293 cells assessed as change in quinpirole-induced intracellular calci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed