Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Delta-type opioid receptor' and Ligand = 'BDBM21121'
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona Tucson

LigandPNGBDBM21121((2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-N-[(...)
Affinity DataKi:  0.360nM ΔG°:  -53.9kJ/mole EC50:  0.770nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona Tucson

LigandPNGBDBM21121((2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-N-[(...)
Affinity DataKi:  0.360nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM21121((2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-N-[(...)
Affinity DataIC50:  1.80nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona Tucson

LigandPNGBDBM21121((2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-N-[(...)
Affinity DataEC50:  0.770nMAssay Description:Agonist activity at human delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed